WAY-100635 maleate

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.

WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor; completely prevents not only the hyperpolarization, with an IC50 of 1.3 nM, but also the decrease in membrane input resistance produced by 5-HT and 5-carboxamidotryptamine with IC50 of 22.5 μM and 50 nM, respectively.Anxiety Phase 1 Discontinued

WAY 100635 maleate salt;WAY100635 maleate salt

Endocrinology/Hormones

5-HT Receptor

5-HT1A

Neurological Disease

Anxiety

634908-75-1

538.64

C29H38N4O6

>98% (HPLC)

DMSO: ≥ 34 mg/mL

COC1=CC=CC=C1N2CCN(CC2)CCN(C3=CC=CC=N3)C(=O)C4CCCCC4.C(=CC(=O)O)C(=O)O

Cyclohexanecarboxamide, N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl-, (2Z)-2-butenedioate (9CI)

(-20℃)

With Ice Pack

≥ 2 years